Synthesis and SAR of highly potent and selective dopamine D 3-receptor antagonists: variations on the 1H-pyrimidin-2-one theme

H Geneste, W Amberg, G Backfisch…

文献索引：Bioorganic and Medicinal Chemistry Letters, , vol. 16, # 7 p. 1934 - 1937

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被引用次数: 22

摘要

... Bioorganic & Medicinal Chemistry Letters. Volume 16, Issue 7, 1 April 2006, Pages 1934–1937. ... Chemical diversity was increased using parallel synthesis (exemplified by compounds 17–22), whereby the intermediate p-nitrophenylcarbamate of amine 1 was generated in situ ...