Novel potent and selective calcium-release-activated calcium (CRAC) channel inhibitors. Part 1: synthesis and inhibitory activity of 5-(1-methyl-3-trifluoromethyl-1H- …
Y Yonetoku, H Kubota, Y Okamoto, A Toyoshima…
文献索引：Bioorganic and Medicinal Chemistry, , vol. 14, # 14 p. 4750 - 4760
... Bioorganic & Medicinal Chemistry. ... To find potent and selective CRAC channel inhibitors, we screened our chemical library and identified N-(4-chlorophenyl)-5-(1-methyl-3-trifluoromethyl- 1H-pyrazol-5-yl)-2-thiophenecarboxamide (4, 10 Fig. 1) as a lead compound. ...
