Formylation en serie arylpyrrolique

JP Boukou-Poba, M Farnier…

文献索引：Boukou-Poba, Jean-Paul; Farnier, Michel; Guilard, Roger Canadian Journal of Chemistry, 1981 , vol. 59, p. 2962 - 2967

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被引用次数: 11

摘要

The formylation of 2-arylpyrroles and methyl 5-arylpyrrole-2-carboxylates (with aryl= benzyl, 2'-thienyl, 3'-thienyl, 2'-furyl, and 3'-furyl) is performed by the Vilsmeier reaction. The orientation of this electrophilic substitution is discussed. The structure of the aldehydes obtained is established by proton nmr data.

~71%

52707-46-7

2-(2-噻吩基)吡咯

~83%

72078-45-6

5-thiophen-2-yl...

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