New, efficient, selective, and one-pot method for acylation of amines

M Basanagouda, MV Kulkarni…

文献索引：Basanagouda, Mahantesha; Kulkarni, Manohar V.; Kalkhambkar, Raj G.; Kulkarni, Geeta M. Synthetic Communications, 2008 , vol. 38, # 17 p. 2929 - 2940

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被引用次数: 4

摘要

Acylation of amines is an important and routinely utilized method for the protection of amino group transformation in organic synthesis. Despite a number of precedents, new efficient methodologies for acylation are still in demand. A variety of catalysts developed for acylation include Lewis acids such as metal halides, [ 1 1. (a) Ahmad , S. ; Iqbal , J. Cobalt(II) chloride catalysed coupling of thiols and anhydrides: A new and efficient synthesis of thiol esters . Tetrahedron Lett . ...