Synthesis of 3-Aryl-3, 4-dihydroisocoumarins

PP Fu, LE Unruh, DW Miller, LW Huang…

文献索引：Fu; Unruh; Miller; et al. Journal of Organic Chemistry, 1985 , vol. 50, # 8 p. 1259 - 1261

被引用次数: 24

摘要

The use of the o-tolyloxazoline as a common intermediate for the general synthesis of a series of 3-aryl-3, 4-dihydroisocoumarins is described. The synthesis involves three single and convenient steps and provides the products in god yields. The products were characterized by analysis of their mass and high-resolution 500-MHz proton NMR spectral data.

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邻甲基苯甲酰氯

Palladium-mediated ortho-alkylation of 2-aryloxazolines

[Clinet, J. C.; Balavoine, G. Journal of Organometallic Chemistry, 1991 , vol. 405, # 2 p. C29 - C31]