Pd (ii)-catalyzed direct C–H acylation of N-Boc hydrazones with aldehydes: one-pot synthesis of 1, 2-diacylbenzenes

S Sharma, A Kim, J Park, M Kim, JH Kwak…

文献索引：Sharma, Satyasheel; Kim, Aejin; Park, Jihye; Kim, Mirim; Kwak, Jong Hwan; Jung, Young Hoon; Park, Jung Su; Kim, In Su Organic and Biomolecular Chemistry, 2013 , vol. 11, # 45 p. 7869 - 7876

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被引用次数: 15

摘要

A palladium (II)-catalyzed direct acylation of acetophenone N-Boc hydrazones with aldehydes via C–H bond activation is described. This protocol provides direct access to a range of 1, 2-diacylbenzenes, which are useful precursors to construct biologically interesting and pharmaceutically important compounds.