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Discovery of a novel sulfonamide-pyrazolopiperidine series as potent and Efficacious γ-Secretase Inhibitors

MY Xiaocong, AW Konradi, J Smith, YZ Xu…

文献索引:Bioorganic and Medicinal Chemistry Letters, , vol. 20, # 7 p. 2195 - 2199

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被引用次数: 13

摘要

... Bioorganic & Medicinal Chemistry Letters. ... a Department of Medicinal Chemistry, Élan Pharmaceuticals, 800 Gateway Boulevard ... b Department of Process and Analytical Chemistry, Élan Pharmaceuticals, 1000 Gateway Boulevard, South San Francisco, CA 94080, United States; ...