Synlett

Efficient synthesis of 7-substituted or 3, 7-disubstituted 1H-indazoles

B Cottyn, D Vichard, F Terrier, P Nioche, CS Raman

文献索引：Cottyn, Betty; Vichard, Dominique; Terrier, Francois; Nioche, Pierre; Raman Synlett, 2007 , # 8 p. 1203 - 1206

被引用次数: 8

摘要

Abstract This work reports on the synthesis of the novel indazole scaffolds 7-OTf-1H- indazole (trifluoromethanesulfonic acid 1H-indazol-7-yl ester), 7-iodo-1H-indazole and 3- bromo-7-iodo-1H-indazole. These new compounds are potent building blocks in divergent syntheses of indazoles via palladium cross-coupling reactions.

570-24-1

2-甲基-6-硝基苯胺

~94%

~52%

~96%

~77%

Inhibitory effects of a series of 7-substituted-indazoles to...

[Cottyn, Betty; Acher, Francine; Ramassamy, Booma; Alvey, Luke; Lepoivre, Michel; Frapart, Yves; Stuehr, Dennis; Mansuy, Daniel; Boucher, Jean-Luc; Vichard, Dominique Bioorganic and Medicinal Chemistry, 2008 , vol. 16, # 11 p. 5962 - 5973]