Discovery of small molecule antagonists of TRPV1

HK Rami, M Thompson, P Wyman, JC Jerman…

文献索引：Bioorganic and Medicinal Chemistry Letters, , vol. 14, # 14 p. 3631 - 3634

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被引用次数: 69

摘要

... Bioorganic & Medicinal Chemistry Letters. ... We therefore initiated an investigation of the SAR of this urea template using array chemistry and a detailed characterisation of the antagonist properties of this compound versus the acid- and heat-mediated activation of TRPV1 using ...