Tetrahedron letters

Synthetic studies in the β-carboline area new entry into4-substituted and 3, 4-disubstituied β-carbolines

N Fukada, ML Trudell, B Johnson, JM Cook

文献索引：Fukada; Trudell; Johnson; Cook Tetrahedron Letters, 1985 , vol. 26, # 18 p. 2139 - 2142

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被引用次数: 15

摘要

Abstract The [3, 3] sigmatropic rearrangement of the allyl ether 2 to provide 3 represents a new synthetic entry into 3, 4-disubstituted β-carbolines. In keeping with the interest in such substituted β-carbolines, the hydrazine mediated conversion of 4-oxo-tetrahydro β-carboline 1b into 4-amino β-carboline 2b is also described, as well as the analogous reaction in the isoquinoline series.