3-Arylamino-2H-1, 2, 4-benzothiadiazin-5-ol 1, 1-dioxides as novel and selective CXCR2 antagonists

Y Wang, J Busch-Petersen, F Wang, L Ma, W Fu…

文献索引：Wang, Yonghui; Busch-Petersen, Jakob; Wang, Feng; Ma, Lanping; Fu, Wei; Kerns, Jeffrey K.; Jin, Jian; Palovich, Michael R.; Shen, Jing-Kang; Burman, Miriam; Foley, James J.; Schmidt, Dulcie B.; Hunsberger, Gerald E.; Sarau, Henry M.; Widdowson, Katherine L. Bioorganic and Medicinal Chemistry Letters, 2007 , vol. 17, # 14 p. 3864 - 3867

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被引用次数: 19

摘要

Download PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... A series of 3-arylamino-2H-1,2,4-benzothiadiazin-5-ol 1,1-dioxides were prepared and shown to be novel and selective antagonists of the CXCR2 receptor. Synthesis, structure and activity relationships, selectivity, and some developability properties are described.