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Fused bicyclic derivatives of 2, 4-diaminopyrimidine as c-Met inhibitors

LR Weinberg, MS Albom, TS Angeles, J Husten…

文献索引:Bioorganic and Medicinal Chemistry Letters, , vol. 21, # 1 p. 164 - 167

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被引用次数: 14

摘要

... Please enable JavaScript to use all the features on this page. Bioorganic & Medicinal Chemistry Letters. ... The C4-substituent was fixed as 2-amino-3-fluoro-N-methylbenzamide, and medicinal chemistry focused on optimizing the C2-benzazepin-2-one. Table 2. ...