Synthesis of 2, 3, 4, 5-tetrahydro-1, 5-methano-1H-3-benzazepine via oxidative cleavage and reductive amination strategies

PR Brooks, S Caron, JW Coe, KK Ng, RA Singer…

文献索引：Synthesis, , # 11 p. 1755 - 1758

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被引用次数: 14

摘要

... Finally, LiAlH 4 reduction provided 5 in 1.2% yield overall from 1. Described herein are high yielding alternatives to the published synthesis of 5 from benzonorbornadiene. Scheme 1. ... 1980, 21: 177; 11 Abdel-Magid AF. ... Longmei Z. Tangsheng P. Huiyan Z. Yan L. Jingyu SJ Org. ...