Tetrahedron letters

A second-generation cycloaddition approach to 3-acyl-4-hydroxypyridin-2-ones

CFR Jones, CE Dawson, MJ O'Mahony, P Patel

文献索引：Jones, Raymond C. F.; Dawson, Claire E.; O'Mahony, Mary J.; Patel, Pravin Tetrahedron Letters, 1999 , vol. 40, # 21 p. 4085 - 4088

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被引用次数: 11

摘要

Download full text in PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... The 1,3-dipolar cycloaddition of the β-aminonitrile oxide, formed from β-alanine, to the enamine of a β-ketoester affords a 3-(2-aminoalkyl)isoxazole-4-carboxylic ester that is converted via isoxazolo[4,5-c]pyridin-4-ones into 3-acetyl-4-hydroxypyridin-2-ones.

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Synthesis of and tautomerism in 3-acyltetramic acids

[Jones, Raymond C. F.; Bhalay, Gurdip; Carter, Paul A.; Duller, Kathryn A. M.; Dunn, Stephen H. Journal of the Chemical Society, Perkin Transactions 1: Organic and Bio-Organic Chemistry (1972-1999), 1999 , # 7 p. 765 - 776]

Synthesis of 1, 3-dioxin-4-ones and their use in synthesis. ...

[Sato, Masayuki; Yoneda, Naoki; Kaneko, Chikara Chemical & Pharmaceutical Bulletin, 1986 , vol. 34, # 2 p. 621 - 627]