Facile one-pot synthesis of aromatic and heteroaromatic sulfonamides

R Pandya, T Murashima, L Tedeschi…

文献索引：Pandya, Rina; Murashima, Takashi; Tedeschi, Livio; Barrett, Anthony G. M. Journal of Organic Chemistry, 2003 , vol. 68, # 21 p. 8274 - 8276

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被引用次数: 81

摘要

A series of arene and heteroarene sulfonamides were prepared in one vessel from aryl and heteroaryl bromides via conversion into the corresponding Grignard reagents using either magnesium or isopropylmagnesium chloride and subsequent reaction with sulfur dioxide, sulfuryl chloride, and an amine.