1, 2, 4-Triazolo [1, 5-a] quinoxaline as a versatile tool for the design of selective human A3 adenosine receptor antagonists: synthesis, biological evaluation, and …

D Catarzi, V Colotta, F Varano, O Lenzi…

文献索引：Catarzi, Daniela; Cecchi, Lucia; Colotta, Vittoria; Filacchioni, Guido; Melani, Fabrizio Journal of Heterocyclic Chemistry, 1992 , vol. 29, # 5 p. 1161 - 1163

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被引用次数: 41

摘要

A number of 4-oxo-substituted 1, 2, 4-triazolo [1, 5-a] quinoxaline derivatives bearing at position-2 the claimed (hetero) aryl moiety (compounds 1-15) but also a carboxylate group (16-28, 32-36) or a hydrogen atom (29-31) were designed as human A3 (hA3) adenosine