Adenosine A 2A antagonists with potent anti-cataleptic activity

…, H Kobayashi, M Ichimura, J Nakamura, H Kase…

文献索引：Shimada, Junichi; Koike, Nobuaki; Nonaka, Hiromi; Shiozaki, Shizuo; Yanagawa, Koji; Kanda, Tomoyuki; Kobayashi, Hiroyuki; Ichimura, Michio; Nakamura, Joji; Kase, Hiroshi; Suzuki, Fumio Bioorganic and Medicinal Chemistry Letters, 1997 , vol. 7, # 18 p. 2349 - 2352

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被引用次数: 91

摘要

Download full text in PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... Structure-activity relationship of 8-styrylxanthines for in vivo adenosine A 2A antagonism were explored. Diethyl substitution both at the 1- and 3-position was found to dramatically potentiate the anti-cataleptic activity. ... Structure-activity relationships of 8-styrylxanthines for in vivo ...