Tetrahedron letters

Chemoselective N-acylation of amino alcohols promoted by magnesium oxide in aqueous organic solution

DH Kim, HS Rho, JW You, JC Lee

文献索引：Kim, Duck-Hee; Rho, Ho-Sik; You, Jae Won; Lee, Jong Chan Tetrahedron Letters, 2002 , vol. 43, # 2 p. 277 - 279

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被引用次数: 23

摘要

Among a number of amidation methods, condensation of acid chloride with amine has been routinely employed in laboratories. Although this method is highly reactive and successful for the preparation of simple amide, the lack of chemoselectivity limits its uses for the N-acylation