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Synthesis and hypocholesterolemic activity of 6, 7-dihydro-4H-pyrazolo [1, 5-a] pyrrolo [3, 4-d] pyrimidine-5, 8-diones, novel inhibitors of acylCoA: cholesterol O- …

SD Larsen, CH Spilman, FP Bell, DM Dinh…

文献索引:Journal of Medicinal Chemistry, , vol. 34, # 5 p. 1721 - 1727

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被引用次数: 16

摘要

... 0022-2623/91/1834-1721$02.50/0 0 1991 American Chemical Society Page 2. 1722 Journal of Medicinal Chemistry, 1991, Vol. 34, No. 5 Scheme I Larsen et al. 1 base R3X -- 2 0 Table I. Synthesis of 4,5-Dioxopyrrolidine-3-carboxylic Acid, Ethyl Esters 1 ...