N-Amination of unsymmetrically substituted pyrimidines. Synthesis of isomeric N-aminopyrimidones

…, K Wurst, JG Schantl, PS Lobanov, AA Potekhin

文献索引：Bodyagin; Ivanov; Wurst; Schantl; Lobanov; Potekhin Chemistry of Heterocyclic Compounds, 2003 , vol. 39, # 2 p. 195 - 199

全文：HTML全文

被引用次数: 2

摘要

Abstract N-Amination of 6-amino-2-methyl-4-pyrimidone with O-(mesitylenesulfonyl) hydroxylamine leads to the 3-amino derivative. The isomeric 1, 6-diamino-2-methyl-4- pyrimidone was obtained by the N-amination of the O-benzoyl derivative of the initial pyrimidone and removal of the benzoyl protection.