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Endomorphin-1 analogues containing β-proline are μ-opioid receptor agonists and display enhanced enzymatic hydrolysis resistance

G Cardillo, L Gentilucci, AR Qasem…

文献索引:Journal of Medicinal Chemistry, , vol. 45, # 12 p. 2571 - 2578

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被引用次数: 104

摘要

... Journal of Medicinal Chemistry. ... Bologna, 40126-Bologna, Italy. J. Med. Chem. , 2002, 45 (12), pp 2571–2578. DOI: 10.1021/jm011059z. Publication Date (Web): May 9, 2002. Copyright © 2002 American Chemical Society. ...