Tetrahedron letters

N-acyl aziridines-C-acylating agents for the preparation of polyketides

B Lygo

文献索引：Lygo, Barry Tetrahedron Letters, 1994 , vol. 35, # 28 p. 5073 - 5074

全文：HTML全文

被引用次数: 6

摘要

Abstract A one-pot synthesis of N-acylaziridines from carboxylic acids has been developed, and their reaction with dianions derived from β-ketoesters studied. The aziridines were found to be efficient C-acylating agents, giving polyketide-like products in good overall