Bulky N-Substituted 1, 3-Benzazaphospholes: Access via Pd-Catalyzed C− N and C− P Cross Coupling, Lithiation, and Conversion to Novel P C− P t Bu2 Hybrid …

…, MK Kindermann, PG Jones, I Dix, J Heinicke

文献索引：Heinicke, J.; Nietzschmann, E.; Tzschach, A. Journal fuer Praktische Chemie (Leipzig), 1983 , vol. 325, # 3 p. 511 - 516

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被引用次数: 51

摘要

We recently reported a convenient access to 1H-1,3-benzazaphospholes by reductive cyclization of 2-phosphonoanilides, but N-substituted derivatives have so far been obtained only by multistep procedures starting with dilithiation of N-methyl-2-bromoaniline.(14) N-Alkylation, a convenient

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Synthese und umlagerungsreaktionen von o-funktionellen pheny...

[Heinicke, J.; Nietzschmann, E.; Tzschach, A. Journal of Organometallic Chemistry, 1983 , vol. 243, # 1 p. 1 - 8]