2, 3-Dihydro-2-oxo-1 H-benzimidazole-1-carboxamides with Selective Affinity for the 5-HT4 Receptor: Synthesis and Structure-Affinity and Structure-Activity …

I Tapia, L Alonso-Cires…

文献索引：Journal of Medicinal Chemistry, , vol. 42, # 15 p. 2870 - 2880

被引用次数: 42

摘要

... Journal of Medicinal Chemistry. ... Chemistry. 2,3-Dihydro-2-oxo-1H-benzimidazole-1- carboxamides 1−10 were prepared by using 2,3-dihydro-2-oxo-1H-benzimidazoles 13 and appropriate aminoalkylpiperazines 18 as key intermediates (Schemes 1−3). ...

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2-羟基苯并咪唑

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Synthesis of 1??alkyl and 1, 3??dialkyl??2??benzimidazolones...

[Journal of Heterocyclic Chemistry, , vol. 18, p. 85 - 89]