Synthesis

Synthesis of β-Carbolines from 2-Acyl-1-benzenesulfonyl-3-iodo-1H-indoles

G Abbiati, EM Beccalli, A Marchesini, E Rossi

文献索引：Abbiati; Beccalli; Marchesini; Rossi Synthesis, 2001 , # 16 p. 2477 - 2483

全文：HTML全文

被引用次数: 26

摘要

Abstract 2-Acyl-1-benzenesulfonyl-3-iodo-1H-indoles and 1-benzenesulfonyl-3-iodo-1H- indole-2-carbaldehyde give in satisfactory yields 1, 3-and 3-substituted-β-carbolines, respectively, by combined palladium-catalyzed coupling with alk-1-ynes followed by 6-endo- dig cycloamination reactions.