Insecticidal and neuroblocking potencies of variants of the imidazolidine moiety of imidacloprid-related neonicotinoids and the relationship to partition coefficient and …

…, R Ishihara, Y Hieda, K Nishimura…

文献索引：Kagabu, Shinzo; Ishihara, Rika; Hieda, Yosuke; Nishimura, Keiichiro; Naruse, Yuji Journal of Agricultural and Food Chemistry, 2007 , vol. 55, # 3 p. 812 - 818

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被引用次数: 52

摘要

The pharmacophore of the neonicotinoid insecticide imidacloprid, nitroiminoimidazolidine, was modified to heterocycles such as thiazolidine, pyrrolidine, dihydroimidazole, dihydrothiazole, and pyridone conjugated to nitroimine (NNO2) or nitromethylene (CHNO2). Their 6-chloro-3-pyridylmethyl or 5-chloro-3-thiazolylmethyl derivatives were examined for insecticidal activity against the American cockroach by injection and for neuroblocking ...