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(E)-Alkenes as replacements of amide bonds: Development of novel and potent acyclic CGRP receptor antagonists

JJ Kim, MR Wood, SJ Stachel, P de Leon…

文献索引:Bioorganic and Medicinal Chemistry Letters, , vol. 24, # 1 p. 258 - 261

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被引用次数: 4

摘要

... Bioorganic & Medicinal Chemistry Letters. Volume 24, Issue 1, 1 January 2014, Pages 258–261. Cover image Cover image. ... a Department of Medicinal Chemistry, Merck & Co., Inc., PO Box 4, 770 Sumneytown Pike, West Point, PA 19486, United States; ...