Selective Fluorescent Nonpeptidic Antagonists For Vasopressin V2 GPCR: Application To Ligand Screening and Oligomerization Assays.

S Loison, M Cottet, H Orcel, H Adihou…

文献索引：Journal of Medicinal Chemistry, , vol. 55, # 20 p. 8588 - 8602

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被引用次数: 21

摘要

... Journal of Medicinal Chemistry. ... G protein-coupled receptors (GPCRs) constitute the largest family of transmembrane signaling molecules in the human genome and represent the most important class of therapeutic targets to the pharmaceutical industry.(1-3) It is of importance ...