Synthesis

The palladium-catalyzed preparation of condensed tetracyclic heterocycles and their application to the synthesis of rac-mangochinine

Z Vincze, AB Bíró, M Csékei, G Timári, A Kotschy

文献索引：Vincze, Zoltan; Biro, A. Beatrix; Csekei, Marton; Timari, Geza; Kotschy, Andras Synthesis, 2006 , # 8 p. 1375 - 1385

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被引用次数: 23

摘要

Abstract Dihydroisoquinoline derivatives and their analogues, prepared by the Bischler- Napieralsky reaction, were converted to their indole-fused derivatives. Scope and limitations of the palladium-catalyzed reaction, proceeding through the tautomeric enamine forms of these compounds, were studied and the process was extended to the preparation of racemic mangochinine.