ICI 174,864

Modify Date: 2024-02-04 11:14:02

ICI 174,864 Structure
ICI 174,864 structure
Common Name ICI 174,864
CAS Number 89352-67-0 Molecular Weight 606.75
Density 1.16 g/cm3 Boiling Point 892.7ºC at 760 mmHg
Molecular Formula C34H46N4O6 Melting Point N/A
MSDS N/A Flash Point 493.7ºC

 Use of ICI 174,864


ICI 174864 is a highly selective, potent δ-receptor antagonist. ICI 174864 is equipotent with naloxone and can not reverse the effect of the μ-agonist [D-Ala2, MePhe4, Gly-Ol5]enkephalin or the κ-agonist tifluadom[1].

 Names

Name ici 174,864
Synonym More Synonyms

 ICI 174,864 Biological Activity

Description ICI 174864 is a highly selective, potent δ-receptor antagonist. ICI 174864 is equipotent with naloxone and can not reverse the effect of the μ-agonist [D-Ala2, MePhe4, Gly-Ol5]enkephalin or the κ-agonist tifluadom[1].
Related Catalog
References

[1]. R Cotton, et, al. ICI 174864: a highly selective antagonist for the opioid delta-receptor. Eur J Pharmacol. 1984, 97,3.  

 Chemical & Physical Properties

Density 1.16 g/cm3
Boiling Point 892.7ºC at 760 mmHg
Molecular Formula C34H46N4O6
Molecular Weight 606.75
Flash Point 493.7ºC
Exact Mass 691.39400
PSA 177.17000
LogP 4.67350
Index of Refraction 1.564

 Synonyms

N,N-DIALLYL-TYR-AIB-AIB-PHE-LEU
Antalarmin hydrochloride
N,N-Diallyl-Tyr-aib-Phe-Leu
L-Leucine,N,N-di-2-propenyl-L-tyrosyl-2-methylalanyl-L-phenylalanyl