GS-626510

Modify Date: 2024-01-10 20:15:11

GS-626510 structure	Common Name	GS-626510
	CAS Number	1637770-13-8	Molecular Weight	394.47
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₂₅H₂₂N₄O	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Use of GS-626510

GS-626510 is a potent, and orally bioavailable BET family bromodomains inhibitor, with Kd values of 0.59-3.2 nM for BRD2/3/4, with IC50 values of 83 nM and 78 nM foe BD1 and BD2, respectively[1].

Name	GS-626510

Description	GS-626510 is a potent, and orally bioavailable BET family bromodomains inhibitor, with Kd values of 0.59-3.2 nM for BRD2/3/4, with IC50 values of 83 nM and 78 nM foe BD1 and BD2, respectively[1].
Related Catalog	Research Areas >> Cancer Signaling Pathways >> Epigenetics >> Epigenetic Reader Domain
Target	BRD2:0.59-2.5 nM (Kd) BRD3:0.65-0.66 nM (Kd) BRD4:1.3-3.2 nM (Kd) BD1:83 nM (IC50) BD2:78 nM (IC50)
References	[1]. Sperandio D, et al. Structure-guided discovery of a novel, potent, and orally bioavailable 3,5-dimethylisoxazole aryl-benzimidazole BET bromodomain inhibitor. Bioorg Med Chem. 2019 Feb 1;27(3):457-469.

Molecular Formula	C₂₅H₂₂N₄O
Molecular Weight	394.47

DC Chemicals Limited
China
Product Name: GS-626510
Price: $Inquiry/100mg $Inquiry/250mg $Inquiry/500mg
Purity: 98.0%
Stocking Period: 3 Day
Contact: Tony Cao

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Chemical & Physical Properties