KB-0742 dihydrochloride
Names
[ CAS No. ]:
2416874-75-2
[ Name ]:
KB-0742 dihydrochloride
Biological Activity
[Description]:
KB-0742 dihydrochloride is a potent, selective and orally active CDK9 inhibitor with an IC50 of 6 nM for CDK9/cyclin T1. KB-0742 dihydrochloride is selective for CDK9/cyclin T1 with >50-fold selectivity over other CDK kinases. KB-0742 dihydrochloride has potent anti-tumor activity.
Chemical & Physical Properties
[ Molecular Formula ]:
C16H27Cl2N5
[ Molecular Weight ]:
360.33