SRI-29329
Names
[ CAS No. ]:
2086809-58-5
[ Name ]:
SRI-29329
Biological Activity
[Description]:
A potent, specific CDC-like kinase (CLK) inhibitor with IC50 of 78, 16 and 86 nM for CLK1, 2 and4, respectively; shows no significant activity for CLK3, CDK1, CDK4 and CDK6 (IC50>1,000 nM).
[References]
References 1. Shi Y, et al. Bioorg Med Chem Lett. 2017 Feb 1;27(3):406-412. View Related Products by Target Cdc2-like Kinase (CLK)
Chemical & Physical Properties
[ Molecular Formula ]:
C20H26ClN7
[ Molecular Weight ]:
399.927