IACS-7e
Names
[ CAS No. ]:
1800477-13-7
[ Name ]:
IACS-7e
Biological Activity
[Description]:
IACS-7e is a potent TRIM24 bromodomain inhibitor with IC50 of 217.8 nM (TRIM24 ligand displacement).
[References]
References 1. Gechijian LN, et al. Nat Chem Biol. 2018 Mar 5. doi: 10.1038/s41589-018-0010-y. View Related Products by Target Bromodomain
Chemical & Physical Properties
[ Molecular Formula ]:
C26H29N3O7S
[ Molecular Weight ]:
527.592