TNKS1/2-IN-1

Names

[ CAS No. ]:
1498300-31-4

[ Name ]:
TNKS1/2-IN-1

Biological Activity

[Description]:

TNKS1/2-IN-1 is a potent tankyrase TNKS1/2 inhibitor with pIC50s ranging from 7.1-8.2. TNKS1/2-IN-1 can be used for research of cancer, fibrosis, and other hyperproliferative diseases[1].

[Related Catalog]:

Research Areas >> Cancer
Signaling Pathways >> Others >> Others

[Target]

TNKS1/2[1]


[References]

[1]. Keenan Richard M, et al. Preparation of quinazolinediones as tankyrase inhibitors for the treatment of cancer: World Intellectual Property Organization, WO2013177349 A2 2013-11-28.

Chemical & Physical Properties

[ Molecular Formula ]:
C26H23F4N3O4

[ Molecular Weight ]:
517.47

Related Compounds