K-(D-1-Nal)-FwLL-NH2
Names
[ CAS No. ]:
1394288-22-2
[ Name ]:
K-(D-1-Nal)-FwLL-NH2
Biological Activity
[Description]:
K-(D-1-Nal)-FwLL-NH2 is a high affinity and potent ghrelin receptor inverse agonist (Ki values are 4.9 and 31 nM in COS7 and HEK293T cells, respectively). K-(D-1-Nal)-FwLL-NH2 blocks ghrelin receptor-mediated Gq- and G13-dependent signaling pathways.
[Related Catalog]:
Chemical & Physical Properties
[ Molecular Formula ]:
C51H67N9O6
[ Molecular Weight ]:
902.13