Lei-Dab 7 TFA
Names
[ CAS No. ]:
1061556-49-7
[ Name ]:
Lei-Dab 7 TFA
Biological Activity
[Description]:
Lei-Dab7 is a high affinity, selective KCa2.2 (SK2) channel blocker (Kd=3.8 nM). Lei-Dab7 exhibits >200-fold selectivity for KCa2.2 over KCa2.1, KCa2.3, KCa3.1, Kv and Kir2.1. Lei-Dab7 increases theta-burst responses and increases LTP in rat hippocampal slices in vitro.
[Related Catalog]:
Chemical & Physical Properties
[ Molecular Formula ]:
C141H236N46O39S6
[ Molecular Weight ]:
3394.07