α-甲基血清素马来酸盐

α-甲基血清素马来酸盐用途

α-methyl Serotonin (maleate) is an agonist of serotonin (5-HT) receptors. It binds selectively to 5-HT1A, 5-HT1B, 5-HT1C, and 5-HT1D receptors over 5-HT1E receptors. It is also selective for 5-HT2B and 5-HT2C receptors over 5-HT2A receptors. α-methyl Serotonin potentiates motor neuron depolarizations induced by NMDA in the presence of the NMDA receptor antagonist memantine. It also increases dopamine release in a dose-dependent manner. α-methyl Serotonin increases systolic blood pressure and transiently increases heart rate.

α-甲基血清素马来酸盐名称

[ CAS 号 ]:
97469-12-0

[ 中文名 ]:
5-羟色胺马来酸α-甲酯

[ 英文名 ]:
α-Me-5-HT

[英文别名 ]:

|A-Methylserotonin maleate salt
2-methyl-5-HT
HMS3262F07

α-甲基血清素马来酸盐物理化学性质

[ 熔点 ]:
191 - 193 °C

[ 分子式 ]:
C₁₅H₁₈N₂O₅

[ 分子量 ]:
306.31400

[ 精确质量 ]:
306.12200

[ PSA ]:
136.64000

[ LogP ]:
2.17530

[ 外观性状 ]:
白色米色粉末

[ 储存条件 ]:
20°C

α-甲基血清素马来酸盐MSDS

详细MSDS(安全技术说明书)

α-甲基血清素马来酸盐安全信息

[ 个人防护装备 ]:
Eyeshields;Gloves;type N95 (US);type P1 (EN143) respirator filter

[ 危险品运输编码 ]:
NONH for all modes of transport

[ 海关编码 ]:
2933990090

α-甲基血清素马来酸盐海关

[ 海关编码 ]: 2933990090

[ 中文概述 ]:
2933990090. 其他仅含氮杂原子的杂环化合物. 增值税率:17.0%. 退税率:13.0%. 监管条件:无. 最惠国关税:6.5%. 普通关税:20.0%

[ 申报要素 ]: 品名, 成分含量, 用途, 乌洛托品请注明外观, 6－己内酰胺请注明外观, 签约日期

[ Summary ]:
2933990090. heterocyclic compounds with nitrogen hetero-atom(s) only. VAT:17.0%. Tax rebate rate:13.0%. . MFN tariff:6.5%. General tariff:20.0%

α-甲基血清素马来酸盐文献

5-HT1 and 5-HT2 binding profiles of the serotonergic agents alpha-methylserotonin and 2-methylserotonin.

J. Med. Chem. 33 , 755-758, (1990)

alpha-Methyl-5-hydroxytryptamine (alpha-Me-5-HT; 2) and 2-methyl-5-hydroxytryptamine (2-Me-5-HT; 3) are considered to be 5-HT2-selective and 5-HT3-selective agents, respectively. These agents were syn...

Serotonin via 5-HT1B and 5-HT2B receptors stimulates anion secretion in the rat epididymal epithelium.

J. Physiol. 519 , 519, (1999)

1. The short-circuit current (Isc) technique was used to study the role of 5-hydroxytryptamine (5-HT) in the regulation of anion secretion in cultured rat cauda epididymal epithelia. 2. 5-HT, the 5-HT...

Effects of serotonin-1 and serotonin-2 receptor agonists on neuronal activity in the nucleus tractus solitarius.

J. Auton. Nerv. Syst. 56 , 119-124, (1995)

Spontaneous neuronal activity in the solitary tract nucleus was recorded extracellularly in a brain slice preparation during bath-application of 5-HT1 and 5-HT2 receptor-selective agonists and antagon...

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α-甲基血清素马来酸盐

α-甲基血清素马来酸盐用途

α-甲基血清素马来酸盐名称

α-甲基血清素马来酸盐物理化学性质

α-甲基血清素马来酸盐MSDS

详细MSDS(安全技术说明书)

α-甲基血清素马来酸盐安全信息

α-甲基血清素马来酸盐海关

α-甲基血清素马来酸盐文献

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α-甲基血清素 马来酸盐

α-甲基血清素 马来酸盐用途

α-甲基血清素 马来酸盐名称

α-甲基血清素 马来酸盐物理化学性质

α-甲基血清素 马来酸盐MSDS

详细MSDS(安全技术说明书)

α-甲基血清素 马来酸盐安全信息

α-甲基血清素 马来酸盐海关

α-甲基血清素 马来酸盐文献

推荐生产厂家/供应商：

热门化合物

α-甲基血清素马来酸盐

α-甲基血清素马来酸盐用途

α-甲基血清素马来酸盐名称

α-甲基血清素马来酸盐物理化学性质

α-甲基血清素马来酸盐MSDS

α-甲基血清素马来酸盐安全信息

α-甲基血清素马来酸盐海关

α-甲基血清素马来酸盐文献