WAY-100635 Maleate
Modify Date: 2024-01-08 11:14:24
WAY-100635 Maleate structure
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Common Name | WAY-100635 Maleate | ||
|---|---|---|---|---|
| CAS Number | 1092679-51-0 | Molecular Weight | 538.635 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C29H38N4O6 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of WAY-100635 MaleateWAY-100635 Maleate is a potent and selective 5-HT1A Receptor antagonist with a pIC50 of 8.87, an apparent pA2 of 9.71. |
| Name | WAY-100635 Maleate |
|---|---|
| Synonym | More Synonyms |
| Description | WAY-100635 Maleate is a potent and selective 5-HT1A Receptor antagonist with a pIC50 of 8.87, an apparent pA2 of 9.71. |
|---|---|
| Related Catalog | |
| Target |
5-HT1A Receptor:8.87 (pIC50) 5-HT1A Receptor:9.71 (pA2) |
| In Vitro | WAY-100635 Maleate is a potent and, at high concentrations, an insurmountable antagonist of the 5-HT1A receptor agonist action of 5-carboxamidotryptamine, with an apparent pA2 value (at 0.3 nM) of 9.71. WAY-100635 displaces specific binding of the 5-HT1A radioligand, [3H]8-OH-DPAT (8-hydroxy-2-(di-n-propylamino)tetralin), to rat hippocampal membranes with a plCIC50 of 8.87[1]. |
| References |
| Molecular Formula | C29H38N4O6 |
|---|---|
| Molecular Weight | 538.635 |
| Exact Mass | 538.279114 |
| PSA | 123.51000 |
| LogP | 3.54040 |
| Cyclohexanecarboxamide, N-[2-[4-(2-methoxyphenyl)-1-piperazinyl]ethyl]-N-2-pyridinyl-, (2Z)-2-butenedioate (1:1) |
| N-{2-[4-(2-Methoxyphenyl)-1-piperazinyl]ethyl}-N-(2-pyridinyl)cyclohexanecarboxamide (2Z)-2-butenedioate (1:1) |
| N-{2-[4-(2-Methoxyphenyl)piperazin-1-yl]ethyl}-N-(pyridin-2-yl)cyclohexanecarboxamide (2Z)-but-2-enedioate (1:1) |
| Cyclohexanecarboxamide (N-[2-[4-(2-methoxyphenyl)-1-piperazinyl]ethyl]-N-2-pyridinyl |
| WAY100635 |