Name | Thrombin inhibitor 1 |
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Description | Thrombin inhibitor 1 is a potent thrombin inhibitor (Ki=0.66 nM, 2xaPTT=0.43 μM). |
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Related Catalog | |
Target |
Ki: 0.66 nM (thrombin)[1] |
In Vitro | Thrombin inhibitor 1 (Compound 4) is binds in the active site of thrombin with Ki of 0.66 nM, 2xaPTT=0.43 uM). Thrombin inhibitor 1 (Compound 4) is evaluated for its thrombin inhibitory potency and its functional ability to double the activated partial thromboplastin time (2xaPTT) in human plasma with a 2xaPTT of 0.43 μM[1]. |
References |
Molecular Formula | C22H20Cl2F2N4O3 |
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Molecular Weight | 497.32 |