ERK1/2 inhibitor 9
Modify Date: 2024-01-16 22:11:37
ERK1/2 inhibitor 9 structure
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Common Name | ERK1/2 inhibitor 9 | ||
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| CAS Number | 2169302-75-2 | Molecular Weight | 586.08 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C31H32ClN7O3 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of ERK1/2 inhibitor 9ERK1/2 inhibitor 9 (Probe 1) is a covalent ERK1/2 inhibitor. ERK1/2 inhibitor 9 shows sub-micromolar activity in cells (A375 GI50=0.47 μM). ERK1/2 inhibitor 9 causes the downregulation of phospho-ERK1/2. ERK1/2 inhibitor 9 tagged trans-cyclo-octene (TCO) and Tz-Thalidomide (tetrazine tagged Thalidomide) can form the corresponding ERK-CLIPTAC to elicit degradation of ERK1/2[1]. |
| Name | ERK1/2 inhibitor 9 |
|---|
| Description | ERK1/2 inhibitor 9 (Probe 1) is a covalent ERK1/2 inhibitor. ERK1/2 inhibitor 9 shows sub-micromolar activity in cells (A375 GI50=0.47 μM). ERK1/2 inhibitor 9 causes the downregulation of phospho-ERK1/2. ERK1/2 inhibitor 9 tagged trans-cyclo-octene (TCO) and Tz-Thalidomide (tetrazine tagged Thalidomide) can form the corresponding ERK-CLIPTAC to elicit degradation of ERK1/2[1]. |
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| Related Catalog | |
| Target |
ERK1 ERK2 |
| References |
| Molecular Formula | C31H32ClN7O3 |
|---|---|
| Molecular Weight | 586.08 |