FR 901537

Modify Date: 2024-03-01 13:05:26

FR 901537 Structure
FR 901537 structure
Common Name FR 901537
CAS Number 161162-21-6 Molecular Weight 507.62300
Density 1.45g/cm3 Boiling Point 897.3ºC at 760 mmHg
Molecular Formula C23H29N3O6S2 Melting Point N/A
MSDS N/A Flash Point 496.5ºC

 Use of FR 901537


FR 901537 is a potent and competitive aromatase inhibitor. FR 901537, a novel naphthol derivative, has the potential for breast cancer research[1].

 Names

Name (2R)-2,4-dihydroxy-N-[3-[2-[(6-hydroxy-2-oxo-1H-benzo[f][1,4]benzothiazin-5-yl)sulfanyl]ethylamino]-3-oxopropyl]-3,3-dimethylbutanamide

 FR 901537 Biological Activity

Description FR 901537 is a potent and competitive aromatase inhibitor. FR 901537, a novel naphthol derivative, has the potential for breast cancer research[1].
Related Catalog
References

[1]. N Oohata, et al. A new aromatase inhibitor, FR901537. I. Taxonomy, fermentation, isolation, physiochemical characteristics and biological activities. J Antibiot (Tokyo). 1995 Aug;48(8):757-62.  

 Chemical & Physical Properties

Density 1.45g/cm3
Boiling Point 897.3ºC at 760 mmHg
Molecular Formula C23H29N3O6S2
Molecular Weight 507.62300
Flash Point 496.5ºC
Exact Mass 507.15000
PSA 209.06000
LogP 3.44930
Vapour Pressure 1.25E-34mmHg at 25°C
Index of Refraction 1.694