GT 2016

Modify Date: 2025-08-25 11:43:02

GT 2016 Structure
GT 2016 structure
 Common Name GT 2016
CAS Number 152241-24-2 Molecular Weight 317.46900
Density N/A Boiling Point N/A
Molecular Formula C19H31N3O Melting Point N/A
MSDS N/A Flash Point N/A

 Use of GT 2016


GT-2016 is a potent, selective, and brain penetrant histamine H3 receptor antagonist with a Ki of 43.8 nM. GT-2016 displays selectivity against H1 and H2 receptors, and has non-active against histamine methyltransferase[1].

 Names

Name 5-Cyclohexyl-1-[4-(1H-imidazol-5-yl)-1-piperidinyl]-1-pentanone
Synonym More Synonyms

 GT 2016 Biological Activity

Description GT-2016 is a potent, selective, and brain penetrant histamine H3 receptor antagonist with a Ki of 43.8 nM. GT-2016 displays selectivity against H1 and H2 receptors, and has non-active against histamine methyltransferase[1].
Related Catalog
Target

H3 Receptor:43.8 nM (Ki)

References

[1]. C E Tedford, et al. Pharmacological characterization of GT-2016, a non-thiourea-containing histamine H3 receptor antagonist: in vitro and in vivo studies. J Pharmacol Exp Ther. 1995 Nov;275(2):598-604.

 Chemical & Physical Properties

Molecular Formula C19H31N3O
Molecular Weight 317.46900
Exact Mass 317.24700
PSA 48.99000
LogP 4.19430

 Synonyms

Grifolic acid
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Chemsrc provides GT 2016(CAS#:152241-24-2) MSDS, density, melting point, boiling point, structure, formula, molecular weight etc. Articles of GT 2016 are included as well.>> amp version: GT 2016

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