(R)-OP-1074

(R)-OP-1074 structure	Common Name	(R)-OP-1074
	CAS Number	1443752-77-9	Molecular Weight	457.56
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₂₉H₃₁NO₄	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Use of (R)-OP-1074

(R)-OP-1074 is the inactive isomer of OP-1074 (HY-125263), and can be used as an experimental control. OP-1074 is a pure antiestrogen and a selective ER degrader (PA-SERD), shows specific antiestrogenic activity for ERα and ERβ, inhibits 17β-estradiol (E2)-stimulated transcriptional activity with IC50 of 1.6 and 3.2?nM, respectively[1].

Name	(R)-OP-1074

Description	(R)-OP-1074 is the inactive isomer of OP-1074 (HY-125263), and can be used as an experimental control. OP-1074 is a pure antiestrogen and a selective ER degrader (PA-SERD), shows specific antiestrogenic activity for ERα and ERβ, inhibits 17β-estradiol (E2)-stimulated transcriptional activity with IC50 of 1.6 and 3.2?nM, respectively[1].
Related Catalog	Research Areas >> Cancer Signaling Pathways >> Others >> Others
References	[1]. Fanning SW, et al. Specific stereochemistry of OP-1074 disrupts estrogen receptor alpha helix 12 and confers pure antiestrogenic activity.Nat Commun. 2018 Jun 18;9(1):2368.

Molecular Formula	C₂₉H₃₁NO₄
Molecular Weight	457.56

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(R)-OP-1074

Use of (R)-OP-1074

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(R)-OP-1074 Biological Activity

Chemical & Physical Properties

The content on this webpage is sourced from various professional data sources. If you have any questions or concerns regarding the content, please feel free to contact service1@chemsrc.com.