188589-61-9

188589-61-9 structure

Name: TFM-4AS-1
Chemical Name: N-(2-trifluoromethylphenyl)-3-oxo-4-methyl-4-aza-5α-androst-1-ene-17β-carboxamide
CAS Number: 188589-61-9
Molecular Formula: C₂₇H₃₃F₃N₂O₂
Molecular Weight: 474.56
Catalog: Research Areas Cancer
Create Date: 2017-08-06 19:03:51
Modify Date: 2025-08-23 19:13:01
TFM-4AS-1 is a selective androgen receptor modulator (SARM). TFM-4AS-1 is a potent androgen receptor (AR) ligand with an IC50 of 38 nm. TFM-4AS-1 is also a gene-selective agonist[1].

Name	N-(2-trifluoromethylphenyl)-3-oxo-4-methyl-4-aza-5α-androst-1-ene-17β-carboxamide
Synonyms	DNQX disodium salt

Description	TFM-4AS-1 is a selective androgen receptor modulator (SARM). TFM-4AS-1 is a potent androgen receptor (AR) ligand with an IC50 of 38 nm. TFM-4AS-1 is also a gene-selective agonist[1].
Related Catalog	Research Areas >> Cancer Signaling Pathways >> Others >> Androgen Receptor
References	[1]. Azriel Schmidt, et, al. Identification of Anabolic Selective Androgen Receptor Modulators with Reduced Activities in Reproductive Tissues and Sebaceous Glands. J Biol Chem. 2009, 284,52.

RIDADR	NONH for all modes of transport