| Name | (R)-Benzyl 2-(5-bromo-1H-indole-3-carbonyl)-pyrrolidine-1-carboxylate |
|---|---|
| Synonyms |
(R)-2-(5-bromo-1H-indole-3-carbonyl)-pyrrolidine-1-carboxylic acid benzyl ester
InterMediate of Eletriptan benzyl (2R)-2-[(5-bromo-1H-indole-3-yl)carbonyl]pyrrolidine-1-carboxylate (R)-2-(5-bomo-1H-indole-3-carbonyl)-pyrrolidine-1-carboxylic acid benzyl ester (R)-3-(N-Benzyloxycarbonylpyrrolidin-2-ylcarbonyl)-5-bromo-1H-indole (R)-5-bromo-3-[(1-methyl-2-pyrrolidinyl)methyl]-1H-indole (R)-2-[(5-Bromo-1H-indol-3-yl)carbonyl]-1-pyrrolidinecarboxylic acid benzyl ester (2R)-2-[(5-BroMo-1H-indol-3-yl)carbonyl]-1-pyrrolidinecarboxylic Acid PhenylMethyl Ester (R)-Benzyl 2-(5-bromo-1H-indole-3-carbonyl)pyrrolidine-1-carboxylate 3-(N-benzyloxycarbonylpyrrolidin-2R-ylcarbonyl)-5-bromo-1H-indole |
| Density | 1.505 |
|---|---|
| Boiling Point | 605ºC at 760 mmHg |
| Molecular Formula | C21H19BrN2O3 |
| Molecular Weight | 427.29100 |
| Flash Point | 319.7ºC |
| Exact Mass | 426.05800 |
| PSA | 62.40000 |
| LogP | 4.85220 |
| Vapour Pressure | 1.38E-14mmHg at 25°C |
| Index of Refraction | 1.678 |
| HS Code | 2933990090 |
|---|
|
~72%
143322-56-9 |
| Literature: Slassi, Abdelmalik; Meng, Charles Q.; Dyne, Kerry; Wang, Xin; Lee, David K. H.; Kamboj, Rajender; McCallum, Kirk L.; Mazzocco, Lucy; Rakhit, Suman Medicinal Chemistry Research, 1999 , vol. 9, # 9 p. 668 - 674 |
|
~72%
143322-56-9 |
| Literature: NPS Allelix Corp. Patent: EP944595 B1, 2003 ; Location in patent: Page/Page column 13 ; EP 0944595 B1 |
|
~%
143322-56-9 |
| Literature: WO2010/121673 A1, ; Page/Page column 16-17 ; |
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Detail
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| Literature: US5545644 A1, ; US 5545644 A US5559129 A1, ; US 5559129 A US5559246 A1, ; US 5559246 A US5578612 A1, ; US 5578612 A US5607951 A1, ; US 5607951 A |
|
~%
Detail
|
| Literature: US5545644 A1, ; US 5545644 A |
|
~%
143322-56-9 |
| Literature: Bioorganic and Medicinal Chemistry Letters, , vol. 13, # 20 p. 3419 - 3421 |
| Precursor 7 | |
|---|---|
| DownStream 3 | |
| HS Code | 2933990090 |
|---|---|
| Summary | 2933990090. heterocyclic compounds with nitrogen hetero-atom(s) only. VAT:17.0%. Tax rebate rate:13.0%. . MFN tariff:6.5%. General tariff:20.0% |