| Name | Somatostatin Antagonist |
|---|---|
| Synonyms |
Cyclosomatostatin
C[AMINOHEPTANOYL-PHE-DTRP-LYS-THR: BZL] 6-(4-aminobutyl)-12-benzyl-9-(1H-indol-3-ylmethyl)-3-(1-phenylmethoxyethyl)-1,4,7,10,13-pentazacycloicosane-2,5,8,11,14-pentone Cyclo(7-Aminoheptanoyl-Phe-D-Trp-Lys-Thr[Bzl]) |
| Description | Cyclosomatostatin is a potent somatostatin (SST) receptor antagonist. Cyclosomatostatin can inhibit somatostatin receptor type 1 (SSTR1) signaling and decreases cell proliferation, ALDH+ cell population size and sphere-formation in colorectal cancer (CRC) cells[1]. |
|---|---|
| Related Catalog | |
| References |
| Density | 1.147g/cm3 |
|---|---|
| Boiling Point | 1118.4ºC at 760 mmHg |
| Molecular Formula | C44H57N7O6 |
| Molecular Weight | 779.96700 |
| Flash Point | 630.2ºC |
| Exact Mass | 779.43700 |
| PSA | 196.54000 |
| LogP | 6.05120 |
| Index of Refraction | 1.558 |
| Storage condition | -20°C |
| Personal Protective Equipment | Eyeshields;Gloves;type N95 (US);type P1 (EN143) respirator filter |
|---|---|
| RIDADR | NONH for all modes of transport |
| WGK Germany | 3 |