Literature: Xu, Zhenrong; Tice, Colin M.; Zhao, Wei; Cacatian, Salvacion; Ye, Yuan-Jie; Singh, Suresh B.; Lindblom, Peter; McKeever, Brian M.; Krosky, Paula M.; Kruk, Barbara A.; Berbaum, Jennifer; Harrison, Richard K.; Johnson, Judith A.; Bukhtiyarov, Yuri; Panemangalore, Reshma; Scott, Boyd B.; Zhao, Yi; Bruno, Joseph G.; Togias, Jennifer; Guo, Joan; Guo, Rong; Carroll, Patrick J.; McGeehan, Gerard M.; Zhuang, Linghang; He, Wei; Claremon, David A. Journal of Medicinal Chemistry, 2011 , vol. 54, # 17 p. 6050 - 6062
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