2929219-77-0

2929219-77-0 structure
2929219-77-0 structure
  • Name: PCSK9-IN-20
  • Chemical Name: PCSK9-IN-20
  • CAS Number: 2929219-77-0
  • Molecular Formula: C27H32N6O5S2
  • Molecular Weight: 584.71
  • Catalog: Signaling Pathways Metabolic Enzyme/Protease Ser/Thr Protease
  • Create Date: 2024-01-08 19:37:19
  • Modify Date: 2024-01-08 19:37:19
  • PCSK9-IN-20 (Compound 3i) is a PCSK9 inhibitor with an IC50 of 3.96 µM. PCSK9-IN-20 decreases PCSK9 and increases LDLR protein expression in vitro[1].

Name PCSK9-IN-20
Description PCSK9-IN-20 (Compound 3i) is a PCSK9 inhibitor with an IC50 of 3.96 µM. PCSK9-IN-20 decreases PCSK9 and increases LDLR protein expression in vitro[1].
Related Catalog
Target

IC50: 3.96 µM (PCSK9)[1]

References

[1]. Zhixin Ma, et al. Identification of benzothiazoles as novel PCSK9 inhibitors. Bioorg Med Chem Lett. 2023 Nov 6:129542.  

Molecular Formula C27H32N6O5S2
Molecular Weight 584.71