502654-40-2
502654-40-2 structure
- Name: CYP4A11/CYP4F2-IN-1
- Chemical Name: CYP4A11/CYP4F2-IN-1
- CAS Number: 502654-40-2
- Molecular Formula: C15H15N3OS
- Molecular Weight: 285.36
- Catalog: Signaling Pathways Metabolic Enzyme/Protease Cytochrome P450
- Create Date: 2022-12-07 12:08:45
- Modify Date: 2024-01-18 10:13:01
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CYP4A11/CYP4F2-IN-1 is a potent dual inhibitor of cytochrome P450 (CYP) 4A11 and CYP4F2, with IC50s of 19 nM and 17 nM, respectively. CYP4A11/CYP4F2-IN-1 has potential for the research of renal diseases[1].
| Name | CYP4A11/CYP4F2-IN-1 |
|---|
| Description | CYP4A11/CYP4F2-IN-1 is a potent dual inhibitor of cytochrome P450 (CYP) 4A11 and CYP4F2, with IC50s of 19 nM and 17 nM, respectively. CYP4A11/CYP4F2-IN-1 has potential for the research of renal diseases[1]. |
|---|---|
| Related Catalog | |
| Target |
CYP4A11:19 nM (IC50) CYP4F2:17 nM (IC50) |
| In Vitro | CYP4A11/CYP4F2-IN-1 (compound 2) inhibits 20-Hydroxyeicosatetraenoic acid (20-HETE) production from arachidonic acid in human renal microsomes, with an IC50 of 4.2 nM[1]. |
| Molecular Formula | C15H15N3OS |
|---|---|
| Molecular Weight | 285.36 |